In this scientific presentation, Dr. Marc Le Borgne will present diverse chemical works on functionalized azaheterocyclic compounds (e.g. indoles, oxazinocarbazoles, indeno[1,2-b]indoles).
All aspects of medicinal chemistry will be discussed: molecular modeling, drug design, process optimization, drug targeting, biological behavior, pharmacological activity, structure-activity relationship and pharmaco-modulation.
Marc Le Borgne is Professor at Faculté de Pharmacie - Institut des Sciences Pharmaceutiques et Biologiques, Université Claude Bernard Lyon 1, France.