Design and Synthesis of Small Molecules as Potential Therapeutic Agents

In this scientific presentation, Dr. Marc Le Borgne will present diverse chemical works on functionalized azaheterocyclic compounds (e.g. indoles, oxazinocarbazoles, indeno[1,2-b]indoles).

All aspects of medicinal chemistry will be discussed: molecular modeling, drug design, process optimization, drug targeting, biological behavior, pharmacological activity, structure-activity relationship and pharmaco-modulation. 

Marc Le Borgne is Professor at Faculté de Pharmacie - Institut des Sciences Pharmaceutiques et Biologiques, Université Claude Bernard Lyon 1, France.

Publisert 9. des. 2010 10:41